Status:

COMPLETED

Influence of Drug Transporter Expression on the Pharmacokinetics of the HIV Protease Inhibitor Kaletra

Lead Sponsor:

Heidelberg University

Conditions:

Healthy

Pharmacokinetics

Eligibility:

All Genders

18-50 years

Brief Summary

The aim of this study is to determine the pharmacokinetics of Kaletra™ (HIV protease inhibitors lopinavir and ritonavir) in different body compartments and to assess the role of four different drug tr...

Detailed Description

Objective: Measurement of AUC, Cmax, tmax, t1/2 and clearance (Cl) of the protease inhibitor Kaletra™ (lopinavir and ritonavir) each in the plasma of healthy individuals * establish free and total p...

Eligibility Criteria

Inclusion

  • Good state of health

Exclusion

  • Drug treatment with known inhibitors or inducers of cytochrome P450 isozymes or ABC-transporters within the preceding 2 months
  • Any acute or chronic illness
  • Smoking
  • Pregnancy
  • Alcohol or drug abuse

Key Trial Info

Start Date :

January 1 2005

Trial Type :

OBSERVATIONAL

Allocation :

ESTIMATED

End Date :

Estimated Enrollment :

12 Patients enrolled

Trial Details

Trial ID

NCT00176033

Start Date

January 1 2005

Last Update

February 13 2009

Active Locations (1)

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Page 1 of 1 (1 locations)

1

Clinical Research Center, Department of Internal Medicine VI

Heidelberg, Germany, 69120