Status:

COMPLETED

A Study to Assess the Safety and Interaction Between Casopitant and Ketoconazole When Taken By Healthy Adults

Lead Sponsor:

GlaxoSmithKline

Conditions:

Nausea and Vomiting, Chemotherapy-Induced

Eligibility:

All Genders

18-55 years

Phase:

PHASE1

Brief Summary

Casopitant may affect liver enzymes that metabolize ketoconazole. This study is designed to test the safety and the extent of the Casopitant affect on ketoconazole levels in healthy human subjects.

Eligibility Criteria

Inclusion

  • Inclusion criteria:
  • A female subject who is non-childbearing potential or using acceptable contraceptive methods.
  • Adequate organ system functions.
  • Able to swallow and retain oral medication.
  • Subject is able to understand and comply with protocol requirements and instruction and is likely to complete the study.
  • Exclusion Criteria:
  • Current clinically relevant abnormality, medical condition, or circumstance that makes the subject unsuitable for the study per the study doctor.
  • History of drug or other allergy which, in the opinion of the study doctor, contraindicates participation.
  • Use of an investigational drug within 28 days or 5 half-lives.
  • Use of prescription or non-prescription drugs, supplements or vitamins (excluding multivitamins) within 14 days, or 5 half-lives prior to first dose of study medication.
  • Blood donation in excess of 500mL within 56 days prior to dosing or intends to donate within 30 days of the post-treatment follow-up visit.
  • Iron deficiency.
  • Positive stool for occult blood.
  • Female subject who is pregnant or lactating.
  • Male subject who has a history of hypogonadism.
  • Positive urine drug screen.
  • Positive for HIV antibody, hepatitis C antibody or hepatitis B surface antigen.
  • Use of tobacco-containing products within the past 12 months prior to screening.
  • History of drug or alcohol abuse or dependence within 6 months of screening.
  • History or presence of uncontrolled emesis.
  • Presence of active infection.
  • History of cholecystectomy or biliary tract disease.
  • Active peptic ulcer disease (PUD) or a history of PUD of unknown etiology.
  • Any degree of heart failure.
  • Consumption of any food or drink containing grapefruit or grapefruit juice, apple juice, Seville oranges, kumquats, pommelos or vegetables from the mustard green family within 7 days prior to the first dose unless prior approval is received.

Exclusion

    Key Trial Info

    Start Date :

    April 16 2007

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    August 27 2007

    Estimated Enrollment :

    85 Patients enrolled

    Trial Details

    Trial ID

    NCT00460707

    Start Date

    April 16 2007

    End Date

    August 27 2007

    Last Update

    August 3 2017

    Active Locations (3)

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    Page 1 of 1 (3 locations)

    1

    GSK Investigational Site

    Overland Park, Kansas, United States, 66211

    2

    GSK Investigational Site

    Buffalo, New York, United States, 14202

    3

    GSK Investigational Site

    Columbus, Ohio, United States, 43212

    A Study to Assess the Safety and Interaction Between Casopitant and Ketoconazole When Taken By Healthy Adults | DecenTrialz