Status:

TERMINATED

Study Evaluating the Pharmacokinetic Profile of RhuDex® in a Tablet Formulation

Lead Sponsor:

MediGene

Conditions:

Pharmacokinetics

Eligibility:

MALE

18-60 years

Phase:

PHASE1

Brief Summary

RhuDex® (code number AV1142742) is a novel, orally bioavailable, low molecular weight modulator of co-stimulation of T lymphocytes. RhuDex® binds to the protein CD80 (also known as B7-1) on the surfac...

Detailed Description

This is an open-label, non-randomized, monocentric Phase I study to evaluate the pharmacokinetic profile of single-dosed and repeat-dosed RhuDex® using a tablet formulation as well as to assess the ef...

Eligibility Criteria

Inclusion

  • Healthy male subjects between 18 and 60 years at the time of enrolment
  • Subjects who are sexually active must use adequate contraception for the duration of the study from screening until 12 weeks after the last dose.
  • BMI between 18.5 and 29.9 kg/m²
  • Written informed consent
  • Ability to comply with the requirements of the study

Exclusion

  • Acute infection at time of enrolment
  • History of chronic inflammation, chronic infection, other chronic disease, autoimmune disorders (e.g. diabetes mellitus) or cancer
  • Clinically significant abnormal ECG
  • Clinically significant abnormal laboratory values (especially in terms of liver or renal insufficiency)
  • Clinically significant physical findings
  • Major surgery within the last 4 weeks prior to enrolment
  • Organ allograft recipient
  • Concomitant or planned treatment which would interfere with study results
  • Any systemic medical treatment, including over the counter products and dietary supplements such as iodine, fluoride or vitamins, within one week before and during the study course
  • Known allergy against any ingredient of the study medication, meglumine, pantoprazole or bovine milk
  • Participation in an investigational trial within 12 weeks prior to enrolment
  • Systemic intake of immunosuppressive or immunomodulatory medication or vaccination within 30 days prior to enrolment and for the whole study duration
  • Blood loss exceeding 450 mL (including blood donations) within 12 weeks prior to enrolment into the study.
  • Medical history of alcohol or drug abuse within the last 2 years or alcohol consumption greater than 21 units per week.
  • A positive alcohol breath test
  • A positive urine drug screen
  • Smokers who smoke \> 5 cigarettes or 5 cigars per day
  • Presence of hepatitis B surface antigen (HBsAg), hepatitis C antibody (HCV Ab) or HIV-1 or HIV-2 antibodies at screening
  • Subject whose partner is pregnant or lactating

Key Trial Info

Start Date :

May 1 2008

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

August 1 2008

Estimated Enrollment :

12 Patients enrolled

Trial Details

Trial ID

NCT00704119

Start Date

May 1 2008

End Date

August 1 2008

Last Update

March 24 2010

Active Locations (1)

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Page 1 of 1 (1 locations)

1

Charles River Clinical Services Edinburgh Ltd

Edinburgh, Scotland, United Kingdom, EH14 4AP