Status:

UNKNOWN

Capiri-sutent Phase-1 in Advanced Colo-rectal Cancer

Lead Sponsor:

Radboud University Medical Center

Conditions:

Colorectal Cancer

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

The primary objective of this Phase 1 study is to identify the recommended dose of capiri and of sunitinib for combination therapy subsequent phase II trials.

Eligibility Criteria

Inclusion

  • Histological proof of colorectal cancer
  • Patients should have failed one previous line of systemic treatment for advanced disease (and not more than one treatment line), either with fluoropyrimidine monotherapy or in combination with oxaliplatin and/or bevacizumab.
  • No prior treatment with irinotecan or sunitinib
  • Age ≥ 18 years
  • WHO PS 0-1 (see Appendix 3, corresponding with Karnofsky ≥ 70% )
  • Life expectancy ≥ 12 weeks
  • Written informed consent

Exclusion

  • No measurable disease according to RECIST criteria.
  • Prior anti-cancer therapy \< 3 weeks before first dose. For cetuximab \< 30 days or bevacizumab \< 60 days prior to the first dose.
  • Unresolved toxicity \> CTC gr 1 from previous anti-cancer therapy (including radiotherapy) except for alopecia.
  • Inadequate bone marrow function (Hb ≤ 5.6 mmol/L, absolute neutrophil count (ANC) ≤ 1.5 x 109/L, platelets ≤100 x 109/L)
  • renal dysfunction (serum creatinine ≥ 1.5x ULN and glomerular filtration rate ≤ 50 ml/min)
  • Prothrombin time (PT) and activated partial thromboplastin time (APTT) \> 2x ULRR
  • Hepatic dysfunction (serum bilirubin ≥ 1.5x ULN, serum transaminases ≥ 2.5 x ULN)
  • Greater than +1 proteinuria on two consecutive dipsticks taken no less then 2 weeks apart unless urinary protein \< 1,5 g in a 24 Hr period.
  • Pregnant or lactating women
  • History of clinical signs/symptoms of CNS metastases
  • Previous intolerance of fluoropyrimidine therapy, known dihydropyrimidine dehydrogenase (DPD) deficiency. Known hypersensitivity to irinotecan or sunitinib of their excipients.
  • No major surgery \< 4 weeks prior to study entry.
  • No radiotherapy \< 4 weeks prior to study entry except for palliative radiotherapy at focal sites.
  • Any evidence of concurrent severe or uncontrolled disease (i.e. uncontrolled hypertension, congestive heart failure, myocardial infarction \< 6 months, chronic active infection, poorly regulated diabetes mellitus)
  • Any previous significant cardiovascular event during previous fluoropyrimidine therapy (i.e.
  • myocardial ischemia or infarction, arterial thrombosis, pulmonary emboli)
  • Mean Qtc with Bazetts correction \> 470 msec in screening ECG, or a history with familial long QT syndrome
  • Significant haemorrhage (\>30 ml bleeding/episode in the last 3 months) or haemoptysis (\>5 ml fresh blood in previous 4 weeks)
  • History of impairment of gastrointestinal function or -disease that may significantly impair the absorption of oral drugs (i.e. uncontrolled nausea, vomiting, diarrhoea, malabsorption syndrome, bowel obstruction, or inability to swallow tablets)
  • Any psychological, familial, sociological or geographical condition potentially hampering compliance with the study protocol and follow-up schedule; those conditions should be discussed with the patient before registration in the trial
  • Concomitant use medication that may significantly affect hepatic cytochrome P450 drug metabolizing activity by way of enzyme induction or inhibition \< 2 weeks if the first dose and throughout the study period (see Appendix 2)
  • Other concomitant anti-cancer therapy.

Key Trial Info

Start Date :

December 1 2008

Trial Type :

INTERVENTIONAL

Allocation :

ESTIMATED

End Date :

December 1 2012

Estimated Enrollment :

32 Patients enrolled

Trial Details

Trial ID

NCT00777478

Start Date

December 1 2008

End Date

December 1 2012

Last Update

February 3 2012

Active Locations (1)

Enter a location and click search to find clinical trials sorted by distance.

Page 1 of 1 (1 locations)

1

University Medical Center Nijmegen st Radboud

Nijmegen, Gelderland, Netherlands, 6525 GH