Status:

COMPLETED

Safety, Antiviral Activity and PK of MRD of BI 201335 in Chronic Hepatitis C Patients Both Treatment Naive and -Experienced

Lead Sponsor:

Boehringer Ingelheim

Conditions:

Hepatitis C, Chronic

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

This study will investigate safety, antiviral activity, and pharmacokinetics of BI 201335 NA in HCV genotype 1 infected patients treated for 14 days monotherapy followed by BI 201335 NA combination th...

Eligibility Criteria

Inclusion

  • Inclusion criteria:
  • 1a. For treatment-naïve patients: no prior therapy with interferon, peginterferon, or ribavirin for acute or chronic hepatitis C infection
  • 1b. For treatment-experienced patients: confirmed virological failure during or after combination treatment with an approved dose of alfa-2a or alfa-2b peginterferon combined with ribavirin; such patients must have received at least 12 weeks of therapy with a 90 day washout period prior to screening and must have documentation of medical history prior to enrolment in 1220.2 2. Age 18 years or older 3. Signed informed consent form prior to trial participation 4. Male or female with documented hysterectomy or menopausal female with last menstrual period at least 6 months prior to screening 5. Chronic hepatitis C infection of genotype 1, diagnosed by positive HCV serology test (HCV Ab positive) or detectable HCV RNA at least 6 months prior to screening 6. HCV viral load \>= 100,000 IU/mL at screening 7. TSH and T4 within normal limits or adequately controlled thyroid function 8. Histological evidence within 36 months prior to study enrolment of any degree of chronic necroinflammatory activity or the presence of fibrosis (Ishak Grade 1-4 or Metavir Grade 1-3)
  • Exclusion criteria:
  • Patients who have been previously treated with at least one dose of any protease inhibitor for acute or chronic hepatitis C infection
  • Evidence of liver disease due to causes other than chronic HCV infection
  • Positive ELISA for HIV-1 or HIV-2
  • Hepatitis B virus (HBV) infection based on presence of Hbs Ag or HBV DNA
  • Any previous liver biopsy consistent with cirrhosis
  • Decompensated liver diseases as evidenced by ascites, portal hypertension, jaundice or hepatic encephalopathy
  • Haemophilia
  • Hemoglobinopathy (e.g., thalassemia major or sickle cell anemia)
  • Severe pre-existing psychiatric disease
  • Poorly controlled diabetes mellitus
  • Ischaemic heart disease
  • Chronic obstructive airway disease
  • Autoimmune disease; including autoimmune hepatitis
  • History of alcohol abuse within the past 12 months
  • Hyperbilirubinemia (conjugated bilirubin) \>1.5x ULN
  • Alkaline phosphatase \>1.5x ULN
  • ALT and AST levels \>= 5 x ULN
  • Hemoglobin \< 12.0 g/dL for women and \< 13.0 g/dL for men
  • White blood cell count \< 2000 cells/mm3
  • Absolute Neutrophil Count \< 1500 cells/mm3
  • Platelet count \< 100,000 cells/mm3
  • Prothrombin time INR (Institutional Normalized Ratio) prolonged to \> 1.5 x ULN
  • Usage of any investigational drug within 30 days prior to enrolment; or the planned usage of an investigational drug during the course of the current study
  • Known hypersensitivity to study drugs

Exclusion

    Key Trial Info

    Start Date :

    September 1 2007

    Trial Type :

    INTERVENTIONAL

    Allocation :

    ACTUAL

    End Date :

    January 25 2011

    Estimated Enrollment :

    96 Patients enrolled

    Trial Details

    Trial ID

    NCT00793793

    Start Date

    September 1 2007

    End Date

    January 25 2011

    Last Update

    September 5 2018

    Active Locations (16)

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    Page 1 of 4 (16 locations)

    1

    1220.2.10 Boehringer Ingelheim Investigational Site

    San Francisco, California, United States

    2

    1220.2.15 Boehringer Ingelheim Investigational Site

    San Francisco, California, United States

    3

    1220.2.17 Boehringer Ingelheim Investigational Site

    Baltimore, Maryland, United States

    4

    1220.2.11 Boehringer Ingelheim Investigational Site

    New York, New York, United States