Status:

COMPLETED

Safety and Efficacy Study of LB80380 in the Patients With Lamivudine-Refractory Chronic Hepatitis B

Lead Sponsor:

LG Life Sciences

Conditions:

Chronic Hepatitis B

Eligibility:

All Genders

18-65 years

Phase:

PHASE1

PHASE2

Brief Summary

The purpose of the study is to investigate the safety and the antiviral activity of ascending multiple oral doses of LB80380 for 12 weeks in adults with lamivudine-refractory chronic hepatitis B infec...

Detailed Description

LB80380, an oral prodrug, is a promising candidate nucleoside analogue with antiviral activity against wild-type HBV. LB80380 is undergoing clinical development by LG Life Sciences for use in the trea...

Eligibility Criteria

Inclusion

  • Compensated chronic hepatitis B patient
  • Presence of serum HBsAg for more than 6 months.
  • Presence of HBeAg for more than 1 month with compensated liver disease
  • Confirmation of YMDD mutants (M552V, M552I and its related double mutant at L528M) by genotyping of the YMDD motif using line probe assay (INNO-LiPA HBV DR assay)
  • Screening HBV DNA value higher than or equal to 1,000,000 copies/mL (measured by the COBAS Amplicor HBV Monitor™ assay)
  • Screening ALT value between 1.5 and 10 x ULN

Exclusion

  • Co-infection with hepatitis C or D virus (HCV or HDV) or HIV
  • Pregnancy or breast-feeding
  • Previous treatment with nucleoside analogue or any other treatment for HBV except for lamivudine within 6 months prior to study entry
  • Treatment with immunomodulatory agent or corticosteroids within 6 months prior to study entry.
  • De-compensated liver disease
  • Screening alpha-fetoprotein (AFP) value \> 20 ng/mL, and a follow-up ultrasonography performed prior to baseline shows findings indicative of HCC.
  • Presence of anti-HBs at screening

Key Trial Info

Start Date :

March 1 2004

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

December 1 2007

Estimated Enrollment :

65 Patients enrolled

Trial Details

Trial ID

NCT00895596

Start Date

March 1 2004

End Date

December 1 2007

Last Update

May 8 2009

Active Locations (4)

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Page 1 of 1 (4 locations)

1

Queen Mary Hospital

Hong Kong, China

2

Korea University Medical Center

Seoul, South Korea

3

Severance Hospital of Yonsei University

Seoul, South Korea

4

The Catholic University of Korea, Kangnam St. Mary's Hospital

Seoul, South Korea