Status:

UNKNOWN

The Development of Oral Nalbuphine Dosage Form

Lead Sponsor:

Tri-Service General Hospital

Conditions:

Healthy

Eligibility:

All Genders

20-40 years

Phase:

NA

Brief Summary

The purpose of this study is to investigate possible responses to pharmacokinetic properties for nalbuphine oral formulations in healthy volunteers.

Eligibility Criteria

Inclusion

  • Normal healthy adult subjects between 20-40 years of age.
  • Body weight within 80-120% of ideal body weight. Ideal body weight = (height-80)0.7
  • Acceptable medical history and physical examination including:
  • Normal chest X-ray and ECG results within six months prior to Period I dosing.
  • No particular clinical significance in general disease history within two months prior to Period I dosing.
  • Acceptable clinical laboratory determinations without significant deviation from normal values within two months prior to Period I dosing, which includes:
  • AST (SGOT)
  • ALT (SGPT)
  • Gama-GT
  • alkaline phosphatase
  • total bilirubin
  • albumin
  • glucose
  • BUN
  • uric acid
  • creatinine
  • total cholesterol
  • triglyceride(TG)
  • Acceptable hematology within two months prior to the study, which includes hemoglobin, hematocrit, red blood cells, MCV, MCH, MCHC, white blood cells, differential white blood cells and platelets.
  • Acceptable urinalysis within two months prior to the study, which includes pH, blood, glucose and protein.
  • Signed the written informed consent to participate in this study.

Exclusion

  • Recent history of drug or alcohol addiction or abuse.
  • A clinically significant disorder involving the cardiovascular, respiratory, renal, gastrointestinal, immunologic, hematologic, endocrine or neurologic system(s) or psychiatric disease (as determined by the clinical investigator).
  • History of allergic response(s) to nalbuphine or related drugs.
  • History of clinically significant allergies including drug allergies or allergic bronchial asthma.
  • Evidence of chronic or acute infectious diseases.
  • Any clinically significant illness or surgery during the four weeks prior to Period I dosing (as determined by the clinical investigator).
  • Taking any drug known to induce or inhibit hepatic drug metabolism within one month prior to the beginning of the study.
  • Receiving any investigational drug within one month prior to Period I dosing.
  • Taking any prescription medication or any nonprescription medication within two weeks prior to Period I doing.
  • Donating greater than 150 ml of blood within two months prior to Period I dosing or donating plasma (e.g., plasmapheresis) within 14 days prior to Period I dosing. All subjects will be advised not to donate blood for four weeks after completing the study.
  • Consumption of caffeine, xanthine-containing products (i.e., coffee, tea, caffeine-containing sodas, colas and chocolate, etc.) and/or alcohol at least 48 hours prior to days on which dosing is scheduled and during the periods when blood samples are being collected.
  • Any other medical reason as determined by the clinical investigator.
  • Patient is pregnant or breastfeeding. Women of childbearing potential must have a negative urine pregnancy test at Baseline.

Key Trial Info

Start Date :

September 1 2008

Trial Type :

INTERVENTIONAL

Allocation :

ESTIMATED

End Date :

Estimated Enrollment :

60 Patients enrolled

Trial Details

Trial ID

NCT00924079

Start Date

September 1 2008

Last Update

June 19 2009

Active Locations (1)

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Tri-Service General Hospitial

Taipei, Taiwan, 11490