Status:

COMPLETED

Trial of Eflornithine Plus Sulindac in Patients With Familial Adenomatous Polyposis (FAP)

Lead Sponsor:

Cancer Prevention Pharmaceuticals, Inc.

Conditions:

Familial Adenomatous Polyposis

Eligibility:

All Genders

18+ years

Phase:

PHASE3

Brief Summary

The purpose of this randomized, double-blind, Phase III trial is to determine if the combination of eflornithine plus sulindac is superior to sulindac or eflornithine as single agents in delaying time...

Eligibility Criteria

Inclusion

  • Diagnosis of phenotypic classical FAP with disease involvement of the duodenum and/or colon/rectum/pouch.
  • Genotype: Adenomatous polyposis coli (APC) mutation (with or without family history) required
  • Classical FAP Phenotype: 100's to 1,000's of colorectal adenomatous polyps, usually appearing in teenage years
  • Upper gastrointestinal (UGI) endoscopy/ lower gastrointestinal (LGI) endoscopy (proctoscopy/colonoscopy) performed within 30 days of randomization.
  • Patients with an intact colon/rectum, except for clinical polyposis, and prophylactic surgery is being considered as a stratification site.
  • Rectal/pouch polyposis as a stratification site as follows:
  • At least three years since colectomy with ileorectal anastamosis (IRA)/proctocolectomy with pouch, and demonstrating polyposis as defined by Stage 1, 2, 3, of the proposed InSiGHT 2011 Staging System (Appendix B) and summarized as follows:
  • Stage 1: 10-25 polyps, all \< 5 mm Stage 2: 10-25 polyps, at least one \> 1 cm Stage 3: \>25 polyps amenable to complete removal, or any incompletely removed sessile polyp, or any evidence of high grade dysplasia, even if completely removed. \[Note: For staging purposes only.\]
  • For all subjects, any rectal/pouch polyps \> 5 mm must be excised at "baseline".
  • Duodenal polyposis as a stratification site; one or more of the following:
  • Current Spigelman Stage 3 or 4.
  • Prior surgical endoscopic intervention within the past six months for Spigelman Stage 3 or 4 that may have been down staged to Spigelman Stage 1 or 2.
  • Hematopoietic Status (within 30 days prior to randomization):
  • No significant hematologic abnormalities
  • White blood cell count (WBC) at least 3,000/mm3
  • Platelet count at least 100,000/mm3
  • Hemoglobin at least 10.0 g/dL
  • No history of clinical coagulopathy
  • Hepatic Status (within 30 days prior to randomization):
  • Bilirubin no greater than 1.5 times ULN
  • Aspartate aminotransferase (AST) and alanine aminotransferase (ALT) no greater than 1.5 times ULN
  • Alkaline phosphatase no greater than 1.5 times ULN
  • Renal Status (within 30 days prior to randomization):
  • a) Creatinine no greater than 1.5 times ULN
  • Hearing:
  • a) No clinically significant hearing loss, defined in Section 6.2, number 9.
  • If female, neither pregnant nor lactating.
  • Negative pregnancy test if female of child-bearing potential. Fertile patients must use effective contraception\*.
  • Absence of gross blood in stool; red blood on toilet paper only acceptable.
  • No discrete gastric or duodenal ulcer greater than 5 mm within the past year except Helicobacter pylori-related peptic ulcer disease treated with antibiotics.
  • No invasive malignancy within the past 5 years except resected non-melanomatous skin cancer, papillary thyroid cancer, or precancerous cervical dysplasia.
  • No other significant medical or psychiatric problems that would preclude study participation or interfere with capacity to give informed consent.
  • Use of 81-100 mg daily aspirin or up to 700 mg aspirin not more than once a week are eligible.
  • No concurrent warfarin, fluconazole, lithium, Pradaxa® or other direct thrombin inhibitors, Plavix®, cyclosporine, other NSAIDs (such as ibuprofen, aspirin, diflunisal), diuretics (furosemide and thiazides), dimethylsulfoxide (DMSO), methotrexate, probenecid, propoxyphene hydrochloride, Tylenol® (acetaminophen) preparations containing aspirin or cytotoxic chemotherapy drugs.
  • Willingness to forego concurrent use of supplements containing omega-3 fatty acids, corticosteroids, non-steroidal anti-inflammatory drugs or other FAP directed drug therapy.
  • Able to provide informed consent and follow protocol requirements.

Exclusion

  • Prior pelvic irradiation.
  • Patients receiving oral corticosteroids within 30 days of enrollment.
  • Treatment with other investigational agents in the prior 4 weeks.
  • Use of other non-steroidal anti-inflammatory drugs (such as ibuprofen) exceeding 4 days per month, in the prior 6 weeks.
  • Regular use of aspirin in excess of 700 mg per week.
  • Treatment with other FAP directed drug therapy (including sulindac or celecoxib, fish oil) within 12 weeks of study enrollment.
  • Hypersensitivity to cyclooxygenase-2 inhibitors, sulfonamides, NSAIDs, or salicylates; NSAID associated symptoms of gastritis.
  • Patients must not have cardiovascular disease risk factors as defined below:
  • Uncontrolled high blood pressure (systolic blood pressure \> 150 mm Hg
  • Unstable angina
  • History of documented myocardial infarction or cerebrovascular accident
  • New York Heart Association Class III or IV heart failure
  • Known uncontrolled hyperlipidemia defined as LDL-C \>= 190 mg/dL or triglycerides \>= 500 mg/dL
  • Patients with significant hearing loss are not eligible for study participation defined as hearing loss that affects everyday life and/or for which a hearing aid is required.
  • Colon/rectum/pouch with high grade dysplasia or cancer on biopsy or a large polyp (\>1 cm) not amenable to complete removal.
  • Duodenal cancer on biopsy.
  • Intra-abdominal desmoid disease, stage III or IV
  • Inability to provide informed consent.

Key Trial Info

Start Date :

October 1 2013

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

March 1 2019

Estimated Enrollment :

171 Patients enrolled

Trial Details

Trial ID

NCT01483144

Start Date

October 1 2013

End Date

March 1 2019

Last Update

June 8 2021

Active Locations (17)

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Page 1 of 5 (17 locations)

1

University of California San Diego

La Jolla, California, United States, 92093

2

Emory University

Atlanta, Georgia, United States, 30322

3

Dana Farber Cancer Institute

Boston, Massachusetts, United States, 02215

4

University of Michigan

Ann Arbor, Michigan, United States, 48109