Status:

COMPLETED

Nelfinavir as Bortezomib-sensitizing Drug in Patients With Proteasome Inhibitor-nonresponsive Myeloma

Lead Sponsor:

Swiss Cancer Institute

Conditions:

Myeloma

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

Trial objectives: To decide whether the addition of nelfinavir to the approved antimyeloma therapy with bortezomib and dexamethasone has sufficient activity in proteasome inhibitor-resistant myeloma ...

Detailed Description

Trial objectives: To decide whether the addition of nelfinavir to the approved antimyeloma therapy with bortezomib and dexamethasone has sufficient activity in proteasome inhibitor-resistant myeloma ...

Eligibility Criteria

Inclusion

  • Patient must give written informed consent prior to any protocol-specific procedure.
  • Patient was diagnosed with multiple myeloma based on standard IMWG criteria, and has received at least one previous line of chemotherapy.
  • Patient has been exposed to or is intolerant to at least one IMID (thalidomide, lenalidomide, pomalidomide).
  • A therapy with bortezomib in the approved dose and schedule, based on Swissmedic approval (treatment of patients with relapsed/refractory multiple myeloma who have received at least one prior line of therapy), is indicated and intended.
  • Patient is refractory to his/her most recent proteasome inhibitor-containing regimen, based on divers criteria.
  • WHO performance status ≤ 3.
  • Age ≥ 18 years.
  • Adequate hematological values: platelets ≥ 50 x 109/L, hemoglobin ≥ 80 g/L (both may be achieved by transfusion).
  • Adequate hepatic function: bilirubin ≤ 1.5 x ULN (for patients with suspected hemolysis: direct bilirubin ≤ 1.5 x ULN), ALT ≤ 3 x ULN (≤ 5 x ULN if liver infiltration by myeloma suspected, based on imaging results).
  • Calculated creatinine clearance ≥ 15 mL/min, according to the formula of Cockcroft-Gault, see Appendix 1).
  • Women are not breastfeeding. Women with child-bearing potential are using effective contraception (see 9.8), are not pregnant and agree not to become pregnant during participation in the trial and during the 12 months thereafter. A negative pregnancy test before inclusion (within 7 days) into the trial is required for all women with child-bearing potential. Men agree not to father a child during participation in the trial and during 12 months thereafter.
  • Completed baseline QoL questionnaire.

Exclusion

  • Evidence of ongoing uncontrolled systemic infections.
  • History of chronic active HCV or HBV.
  • Evidence of myeloma within the CNS.
  • Psychiatric disorder precluding understanding of information on trial related topics, giving informed consent, filling out quality of life (QoL) forms, or interfering with compliance for oral drug intake.
  • Exposure to another experimental drug within 3 weeks prior to trial entry.
  • Any serious underlying medical condition (at the judgment of the investigator) which may impair the ability of the patient to participate in the trial, in particular any uncontrolled clinically significant active disease (e.g. active autoimmune disease, uncontrolled diabetes, uncontrolled cardiac disease).
  • Non-hematologic active malignancy within the past 5 years with the exception of a) adequately treated basal cell carcinoma, squamous cell skin cancer, or thyroid cancer; b) carcinoma in situ of the cervix or breast; c) prostate cancer of Gleason Grade 6 or less with stable prostate-specific antigen levels; or d) cancer considered cured by surgical resection or unlikely to impact survival during the duration of the study, such as localized transitional cell carcinoma of the bladder or benign tumors of the adrenal or pancreas.
  • Concomitant use of other anti-cancer medication or radiotherapy except for local pain control. The use of bisphosphonates is allowed.
  • Significant neuropathy (Grades 3-4, or Grade 2 with pain) within 14 days prior to enrollment.
  • Known hypersensitivity to bortezomib or nelfinavir or hypersensitivity to components of these drugs.
  • Any psychological, familial, sociological or geographical condition likely hampering compliance with the trial protocol and follow-up.
  • Patient who takes the following drugs during the trial therapy, which cannot be replaced or paused.

Key Trial Info

Start Date :

December 2 2014

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

April 17 2018

Estimated Enrollment :

34 Patients enrolled

Trial Details

Trial ID

NCT02188537

Start Date

December 2 2014

End Date

April 17 2018

Last Update

June 26 2019

Active Locations (12)

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Page 1 of 3 (12 locations)

1

Kantonsspital Aarau

Aarau, Switzerland, CH-5001

2

Kantonsspital Baden

Baden, Switzerland, 5404

3

Universitaetsspital-Basel

Basel, Switzerland, CH-4031

4

Istituto Oncologico Svizzera Italiana IOSI

Bellinzona, Switzerland, 6500