Status:

TERMINATED

Tipranavir and Ritonavir vs. Saquinavir and Ritonavir Used With Two Nucleoside Reverse Transcriptase Inhibitors in Single Protease Inhibitor-experienced HIV-1 Patients

Lead Sponsor:

Boehringer Ingelheim

Conditions:

HIV Infections

Eligibility:

All Genders

18+ years

Phase:

PHASE2

Brief Summary

Objectives of the study were to evaluate the efficacy and safety of two different doses of tipranavir (TPV) in combination with ritonavir (TPV/r) compared with a standard dual PI combination of saquin...

Eligibility Criteria

Inclusion

  • Clinical failure while on the current PI-containing regimen of indinavir, nelfinavir, or amprenavir
  • In the investigator's opinion, adherence to the present PI-containing regimen
  • Exposure of \>=6 months to the current PI therapy
  • Stable PI-containing regimen, i.e., receiving the current two reverse transcriptase inhibitors (RTIs) for at least 2 months prior to study entry
  • HIV-1 RNA \>=1000 copies/mL (assayed using the Amplicor polymerase chain reaction (PCR) method at the initial screening visit)
  • No limit in CD4+ cell count at the initial screening
  • At least two new nucleoside reverse transcriptase inhibitor (NRTI) options available
  • Age \>=18 years
  • Acceptable screening laboratory test values that indicated adequate baseline organ function at the time of screening. Acceptable laboratory test values consisted of the following: severity \<=Grade 1 (ACTG Grading Scale). Stable Grade 2 abnormalities were permitted if the values had been demonstrated and documented for at least \>=2 months. All laboratory values \>Grade 2 were subject to approval by the P\&U Clinical Program Leader or designated personnel and subsequently by the BI designated personnel
  • Acceptable medical history, physical examination, ECG, and chest radiograph prior to entry into the treatment phase of the study
  • Use of a barrier contraceptive method of birth control for at least 30 days prior to study drug administration, during the study, and 30 days after study completion
  • Ability to swallow numerous tablets and capsules without difficulty
  • Ability to understand and provide informed consent. Minors had to have approval of a parent or legal guardian

Exclusion

  • Treatment with more than one PI-containing regimen
  • Clinically significant active or acute (onset within the month previous to study entry) medical problems, including the following: opportunistic infections, e.g., active cryptococcosis, Pneumocystis carinii pneumonia, herpes zoster, histoplasmosis, or cytomegalovirus; nonopportunistic diseases, including but not limited to the following: progressive multifocal leukoencephalopathy, lymphoma, or malignancy requiring systemic therapy
  • Prior exposure (\>7 days) to tipranavir, saquinavir, or ritonavir
  • History of clinically significant nervous system or muscle diseases, seizure disorder, or psychiatric disorder that might impair adherence to the protocol
  • Taking of any known P450 3A enzyme-inducing drugs within 30 days of study entry and including the following: rifabutin, rifampin, carbamazepine, dexamethasone, phenobarbital, phenytoin, sulfadimidine, sulfinpyrazone, or troleandomycin
  • Hypersensitivity to tipranavir, saquinavir, or ritonavir
  • Use of interferons, interleukins, HIV vaccines, or any active immunizations within 30 days of study entry
  • Taking of any investigational medication with the exception of adefovir dipivoxil (Preveon™) within 30 days of study entry
  • Pregnancy or lactation (serum β-human chorionic gonadotrophin test had to have been negative within 14 days of study entry)
  • Evidence of substance abuse, which in the investigator's opinion could affect adherence to the protocol
  • In the investigator's judgment, inability to comply with the protocol requirements for reasons other than those specified

Key Trial Info

Start Date :

December 1 1999

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

Estimated Enrollment :

79 Patients enrolled

Trial Details

Trial ID

NCT02239835

Start Date

December 1 1999

Last Update

September 15 2014

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