Status:

COMPLETED

Study of N91115 in Patients With Cystic Fibrosis Homozygous F508del-CFTR Mutation

Lead Sponsor:

Nivalis Therapeutics, Inc.

Conditions:

Cystic Fibrosis

Eligibility:

All Genders

18-80 years

Phase:

PHASE1

Brief Summary

This Phase 1b study in F508del-CFTR homozygous CF patients is being conducted to assess the safety of N91115 as the sole cystic fibrosis transmembrane conductance regulator (CFTR) modulator at doses n...

Detailed Description

Study procedures, frequency and timing are provided in the attached study schema. Adverse events and concomitant medication will be monitored throughout the study from informed consent signing until e...

Eligibility Criteria

Inclusion

  • Male or female, age ≥ 18 years with confirmed diagnosis of CF, homozygous for the F508del-CFTR mutation based on historical results generated by Ambry Genetics within the past two years or if unavailable, confirmed by testing done within the past 28 days
  • Sweat chloride ≥ 60 (milliequivalents) mEq/L, by quantitative pilocarpine iontophoresis test (QPIT) at screening
  • Weight ≥ 40 kg at screening
  • Forced expiratory volume (FEV1) ≥ 40% of predicted normal for age, gender, and height (Hankinson standards) pre- or post-bronchodilator value, at screening
  • Oxygen saturation by pulse oximetry ≥ 90% breathing ambient air, at screening
  • Hematology, clinical chemistry and urinalysis results with no clinically significant abnormalities that would interfere with the study assessments at screening

Exclusion

  • Any acute infection, including acute upper or lower respiratory infections and pulmonary exacerbations that require treatment or hospitalization within 2 weeks of Study Day 1
  • Any change in chronic therapies for CF lung disease (e.g., Ibuprofen, Pulmozyme®, hypertonic saline, Azithromycin, Tobi®, Cayston®) within 4 weeks of Study Day 1
  • Blood hemoglobin \< 10 g/dL at screening
  • Serum albumin \< 2.5 g/dL at screening
  • Abnormal liver function defined as ≥ 3 x upper limit of normal (ULN) in 3 or more of the following: aspartate aminotransferase (AST), alanine aminotransferase (ALT), g-glutamyl transferase (GGT), alkaline phosphatase (ALP), or total bilirubin at screening
  • History of abnormal renal function (creatinine clearance \< 50 mL/min using Cockcroft-Gault equation) within a year of screening
  • History, including the screening assessment, of ventricular tachycardia or other ventricular arrhythmias
  • History, including the screening assessment, of prolonged cardiac QT interval and/or QTcF (QT with Fridericia's correction) interval (\> 450 msec)
  • History of solid organ or hematological transplantation
  • History of alcohol abuse or drug abuse (including cannabis, cocaine, and opioids) in the year prior to screening
  • Use of continuous (24 hr/day) or nocturnal supplemental oxygen

Key Trial Info

Start Date :

February 1 2015

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

July 1 2015

Estimated Enrollment :

51 Patients enrolled

Trial Details

Trial ID

NCT02275936

Start Date

February 1 2015

End Date

July 1 2015

Last Update

November 7 2016

Active Locations (19)

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Page 1 of 5 (19 locations)

1

University of Alabama @ Birmingham

Birmingham, Alabama, United States, 35294

2

Stanford University

Palo Alto, California, United States, 94304

3

Children's CO

Aurora, Colorado, United States, 80045

4

National Jewish Health

Denver, Colorado, United States, 80206