Status:

COMPLETED

A Study to Evaluate the Effects of Rifampin on Pharmacokinetics (PK) of Pevonedistat in Participants With Advanced Solid Tumors

Lead Sponsor:

Millennium Pharmaceuticals, Inc.

Conditions:

Advanced Solid Neoplasm

Eligibility:

All Genders

18+ years

Phase:

PHASE1

Brief Summary

The purpose of this study is to assess the effect of multiple-dose administration of rifampin on the single dose PK of pevonedistat in adult participants with advanced solid tumors.

Detailed Description

The study will enroll approximately 20 participants. The study will be conducted in two Parts: Part A and optional Part B. Part A will have a drug-drug interaction (DDI) assessment. In Part A, partici...

Eligibility Criteria

Inclusion

  • Adult participants who have a histologically or cytologically confirmed metastatic or locally advanced solid tumor that is appropriate for treatment with either docetaxel or carboplatin + paclitaxel in Part B of this study, or have progressed despite standard therapy, or for whom conventional therapy is not considered effective.
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 to 1.
  • Expected survival of at least 3 months from the date of enrollment in the study.
  • Recovered (that is, less than or equal to (\<=) Grade 1 toxicity) from the effects of prior antineoplastic therapy.
  • Adequate organ functions (kidney, liver, cardiac, bone marrow).
  • Suitable venous access for the study-required blood sampling (including PK sampling).

Exclusion

  • Prior treatment with radiation therapy involving greater than or equal to (\>=) 25% of the hematopoietically active bone marrow.
  • Life-threatening illness or serious (acute or chronic) medical or psychiatric illness unrelated to cancer.
  • Active, uncontrolled infection or severe infectious disease.
  • Known human immunodeficiency virus (HIV) seropositive or known hepatitis B or hepatitis C infection.
  • With significant heart or pulmonary disease.
  • Requiring chronic treatment with breast cancer resistance protein (BCRP) inhibitors.
  • Criteria for Continuation into Optional Part B:
  • To be eligible for Part B, participants must have completed Part A and be reassessed to determine if they meet the continuation criteria for Part B.

Key Trial Info

Start Date :

August 13 2018

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

February 28 2021

Estimated Enrollment :

20 Patients enrolled

Trial Details

Trial ID

NCT03486314

Start Date

August 13 2018

End Date

February 28 2021

Last Update

April 18 2022

Active Locations (4)

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Page 1 of 1 (4 locations)

1

Emory University

Atlanta, Georgia, United States, 30308

2

Robert H. Lurie Comprehensive Cancer Center of Northwestern University

Chicago, Illinois, United States, 60611

3

Barbara Ann Karmanos Cancer Institute

Detroit, Michigan, United States, 48201-2013

4

Greenville Health System - Institute for Translational Oncology Research

Greenville, South Carolina, United States, 29605