Status:

COMPLETED

Relative Bioavailability of CE-Iohexol (Captisol-enabled™ Iohexol) Injection and Omnipaque™ Injection

Lead Sponsor:

CyDex Pharmaceuticals, Inc.

Collaborating Sponsors:

Ligand Pharmaceuticals

Syneos Health

Conditions:

Contrast-induced Nephropathy

Coronary Angiography

Eligibility:

All Genders

18+ years

Phase:

NA

Brief Summary

This study is designed to compare the bioavailability of the test Product(CE-Iohexol Injection) and the reference product Iohexol Injection (Omnipaque™) following intravenous injection in normal healt...

Detailed Description

This is a single center, randomized, double-blind, 2-period, crossover study. A total of 24 subjects will be enrolled in the study; subjects will be dosed as 2 groups of 12 subjects each. Additional s...

Eligibility Criteria

Inclusion

  • Women of childbearing potential who are sexually active with a non-sterile male partner must be using a medically acceptable form of birth control for the duration of the trial and for 30 days after the last dose of study drug
  • BMI within the range of 18.5-35 kg/m2, inclusive, and body weight \> 45 kg
  • No significant disease or abnormal laboratory values
  • Normal vital signs, without any clinically significant abnormalities
  • Normal 12-lead electrocardiogram, without any clinically significant abnormalities of rate, rhythm or conduction
  • Nonsmokers defined as not having smoked in the past 3 months prior to dosing
  • Estimated glomerular filtration rate (eGFR) of \> 60 mL/min/1.73 m2

Exclusion

  • Known hypersensitivity or allergy to iohexol, CAPTISOL®, Omnipaque™ or its excipients
  • Known hypersensitivity or allergy to iodine or radio-opaque dyes
  • Women who are pregnant or breast feeding
  • History or presence of asthma or other pulmonary disease, thyroid disease (hypo- or hyperthyroidism), hepatitis or other liver disease
  • Any disease or condition (medical or surgical) which, in the opinion of the investigator, might compromise a major system; or other conditions that may interfere with the absorption, distribution, metabolism or excretion of study drug, or would place the subject at increased risk
  • Abnormal laboratory values which are considered clinically significant
  • Positive screen for Hepatitis B (HbsAg, Hepatitis B Surface Antigen), Hepatitis C (anti HCV, Hepatitis C Antibody), or HIV (anti-HIV 1/2)
  • Participation in a clinical research study involving the administration of an investigational or marketed drug or device within 30 days prior to the first dose
  • Use of medication other than topical products without significant systemic absorption, hormonal contraceptives and hormone replacement therapy
  • Unwilling to refrain from consumption of alcohol within 48 hours prior to each dose administration and during any in-patient period.
  • Positive urine drug screen, positive alcohol breath test or positive cotinine test at screening and upon check-in to the study facility
  • History of significant alcohol abuse within one year prior to screening or regular use of alcohol within six months prior to the screening visit
  • Illicit drug use,significant mental illness, physical dependence to any opioid, or any history of drug abuse or addiction
  • A history of difficulty with donating blood or with the insertion of large-calibre catheter
  • Donation of plasma (500 mL) within 7 days prior to drug administration.
  • Hemoglobin \< 128 g/L (males) and \< 115 g/L (females) and hematocrit \< 0.36 L/L (males) and \< 0.32 L/L (females) at screening
  • Any history of photosensitivity

Key Trial Info

Start Date :

April 12 2019

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

June 15 2019

Estimated Enrollment :

24 Patients enrolled

Trial Details

Trial ID

NCT03869983

Start Date

April 12 2019

End Date

June 15 2019

Last Update

August 16 2019

Active Locations (1)

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Syneos Health Clinique

Québec, Quebec, Canada, G1P0A2