Status:

TERMINATED

Phase 1/2 Study of OBI-999 in Patients With Advanced Solid Tumors

Lead Sponsor:

OBI Pharma, Inc

Conditions:

Locally Advanced Solid Tumor

Eligibility:

All Genders

18+ years

Phase:

PHASE1

PHASE2

Brief Summary

The purpose of this study is to establish the maximum tolerated dose (MTD) and recommended phase 2 dose (RP2D) of OBI-999 as monotherapy, and to characterize the safety and preliminary clinical activi...

Eligibility Criteria

Inclusion

  • Male or female patients, 18 years of age or older at the time of consent.
  • Provide written informed consent prior to performing any study related procedure.
  • Histologically or cytologically confirmed patients with advanced solid tumors.
  • Patients must have been treated with established standard-of-care therapy, or physicians have determined that such established therapy is not sufficiently efficacious, or patients have declined to receive standard-of-care therapy. In the latter case, the informed consent must state the effective therapies the patient is declining.
  • Measurable disease (i.e., at least one measurable lesion per RECIST 1.1)
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
  • Adequate organ function defined as:
  • a. Hepatic:
  • i. Serum ALT ≤3 × upper limit of normal (ULN), ≤5 × ULN in the presence of liver metastases
  • ii. Serum AST ≤3 × ULN, ≤5 × ULN in presence of liver metastases
  • iii.Serum bilirubin ≤1.5 × ULN (unless due to Gilbert's syndrome or hemolysis)
  • b. Renal:
  • i. Creatinine clearance \>50 mL/minute using Cockcroft Gault equation
  • c. Hematologic:
  • i. Absolute neutrophil count ≥1,500/µL
  • ii. Platelets ≥100,000/µL
  • iii. Hemoglobin ≥8 g/dL
  • Patient is willing and able to comply with all protocol required assessments, visits, and procedures, including a pretreatment tumor biopsy. Archival tumor biopsies are acceptable at baseline.
  • Females of childbearing potential must have negative serum pregnancy test prior to starting study therapy, and agree to use a reliable form of contraceptive during the study treatment period and for at least 120 days following the last dose of study drug.
  • Patient not of childbearing potential (i.e., permanently sterilized, postmenopausal) can be included in study. Postmenopausal is defined as 12 months with no menses without an alternative medical cause.
  • Male patients must agree to use an adequate method of contraception during the study treatment period and for at least 120 days following the last dose of study drug.
  • Cannot be breast feeding.
  • Patients with human immunodeficiency virus (HIV) infection are eligible if CD4+ T cell counts ≥ 350 cells/uL; patients on antiretroviral therapy (ART) should be on an established dose for at least 4 weeks and have an HIV viral load less than 400 copies/mL prior to enrollment.
  • Patients with serological evidence of chronic hepatitis B virus (HBV) infection are eligible if they have an HBV viral load below the limit of quantification with or without concurrent viral suppressive therapy.
  • Patients with a history of hepatitis C virus (HCV) infection should have completed curative antiviral treatment and have a viral load below the limit of quantification.
  • Patients in Part B (Cohort-Expansion) must have documented Globo H H score of at least 100 from a qualified laboratory IHC assay in one of the sponsor-selected tumor types to be enrolled in the respective cohort:
  • Cohort 1: Pancreatic cancer
  • Cohort 2: Esophageal cancer
  • Cohort 3: Gastric cancer
  • Cohort 4: Colorectal cancer
  • Cohort 5: Basket (any solid tumor type other than those included in Cohorts 1 through 4).

Exclusion

  • Less than 3 weeks from prior cytotoxic chemotherapy or radiation therapy; and less than 5 half-lives or 3 weeks, whichever is shorter, from prior biologic therapies, prior to the first dose of OBI 999.
  • Has undergone a major surgical procedure (as defined by the Investigator) or significant traumatic injury within 28 days prior to the first dose of OBI 999.
  • Sensory or motor neuropathy of Grade 2 or greater.
  • Patients with a history of solid organ transplant.
  • Unresolved toxicities from prior anticancer therapy, defined as having not resolved to Grade 0 or 1 (using NCI CTCAE version 5.0), except for alopecia and laboratory values listed in the inclusion criteria.
  • Receipt of any prior therapy targeting Globo H.
  • Known hypersensitivity to OBI 999 or its excipients.
  • Has known untreated central nervous system metastases. Patients with treated brain metastases are eligible if there is no evidence of progression for at least 4 weeks after CNS-directed treatment, as ascertained by clinical examination and brain imaging (magnetic resonance imaging \[MRI\] or computed tomography \[CT\]) during the screening period.
  • Has significant clinical cardiac abnormality (e.g., clinical heart failure or unstable angina)
  • Any medical co morbidity that is life threatening or, in the opinion of the Investigator, renders the patient unsuitable for participation in a clinical trial due to possible noncompliance, would place the patient at an unacceptable risk and/or potential to affect interpretation of results of the study.
  • Is receiving any concurrent prohibited medication

Key Trial Info

Start Date :

November 25 2019

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

October 27 2023

Estimated Enrollment :

44 Patients enrolled

Trial Details

Trial ID

NCT04084366

Start Date

November 25 2019

End Date

October 27 2023

Last Update

March 26 2025

Active Locations (4)

Enter a location and click search to find clinical trials sorted by distance.

Page 1 of 1 (4 locations)

1

Scripps MD Anderson Cancer Center

La Jolla, California, United States, 92037

2

Memorial Sloan Kettering Cancer Center

New York, New York, United States, 10065

3

West Cancer Center

Germantown, Tennessee, United States, 38138

4

University of Texas MD Anderson Cancer Center

Houston, Texas, United States, 77030