Status:

COMPLETED

Effect of BIA 5-1058 on the Steady State Pharmacokinetics of Treprostinil

Lead Sponsor:

Bial - Portela C S.A.

Conditions:

Pulmonary Arterial Hypertension

Eligibility:

All Genders

18-45 years

Phase:

PHASE1

Brief Summary

The purpose of this study is to assess the effect of BIA 5-1058 200 mg on the pharmacokinetic (PK) of treprostinil

Detailed Description

This study was an open-label, three period, fixed sequence study in healthy male and female subjects performed at a single study center. The study comprised: * Screening during Days -28 to -2 (both ...

Eligibility Criteria

Inclusion

  • Provided a signed and dated informed consent before any study specific procedures were conducted.
  • Male and female subjects aged 18 to 45 years (both inclusive) at the Screening Visit.
  • Healthy as determined by the Principal Investigator based on medical history, physical examination, clinical laboratory test results, vital signs and digital 12 lead electrocardiogram (ECG). If a vital sign or ECG assessment was outside of the reference range at the Screening Visit or baseline, the assessment could have been repeated once as soon as possible and in any cases before enrolment to rule out any error.
  • Non-smoker or ex-smoker for at least 3 months prior to the Screening Visit.
  • Body mass index (BMI) between 18.5 and 29.9 kg/m2 (both inclusive) at the Screening Visit and on admission to each treatment period.
  • Negative test results for hepatitis B surface antigen (HBsAg), hepatitis B core antibody (anti HBc), immunoglobulin M (IgM) anti-HBc, hepatitis C virus antibody (anti HCV) and human immunodeficiency virus (HIV) (Types 1 and 2) antibodies at the Screening Visit.
  • Negative screen for alcohol and drugs of abuse at the Screening Visit and on admission to each treatment period.
  • Subject had to be willing and able to be confined to the clinical unit and had to adhere to the study and lifestyle restrictions.
  • Contraception requirements:
  • Male subjects had to use together with his female partner/spouse a highly effective contraception form of birth control in combination with a barrier method throughout the clinical study period and agreed not to father a child or to donate sperm starting at the Screening Visit and throughout the clinical study.
  • Female subjects had to either be of non childbearing potential or had to use highly effective methods of contraception from at least 3 months before the Screening Visit and throughout the clinical study in combination with a barrier method.

Exclusion

  • Inclusion Criteria:
  • Subjects who met the following criteria were considered eligible to participate/continue in the study:
  • Provided a signed and dated informed consent before any study specific procedures were conducted.
  • Male and female subjects aged 18 to 45 years (both inclusive) at the Screening Visit.
  • Healthy as determined by the Principal Investigator based on medical history, physical examination, clinical laboratory test results, vital signs and digital 12 lead electrocardiogram (ECG). If a vital sign or ECG assessment was outside of the reference range at the Screening Visit or baseline, the assessment could have been repeated once as soon as possible and in any cases before enrolment to rule out any error.
  • Non-smoker or ex-smoker for at least 3 months prior to the Screening Visit.
  • Body mass index (BMI) between 18.5 and 29.9 kg/m2 (both inclusive) at the Screening Visit and on admission to each treatment period.
  • Negative test results for hepatitis B surface antigen (HBsAg), hepatitis B core antibody (anti HBc), immunoglobulin M (IgM) anti-HBc, hepatitis C virus antibody (anti HCV) and human immunodeficiency virus (HIV) (Types 1 and 2) antibodies at the Screening Visit.
  • Negative screen for alcohol and drugs of abuse at the Screening Visit and on admission to each treatment period.
  • Subject had to be willing and able to be confined to the clinical unit and had to adhere to the study and lifestyle restrictions.
  • Contraception requirements:
  • Male subjects had to use together with his female partner/spouse a highly effective contraception form of birth control in combination with a barrier method throughout the clinical study period and agreed not to father a child or to donate sperm starting at the Screening Visit and throughout the clinical study.
  • Female subjects had to either be of non childbearing potential or had to use highly effective methods of contraception from at least 3 months before the Screening Visit and throughout the clinical study in combination with a barrier method.

Key Trial Info

Start Date :

February 28 2018

Trial Type :

INTERVENTIONAL

Allocation :

ACTUAL

End Date :

May 25 2018

Estimated Enrollment :

20 Patients enrolled

Trial Details

Trial ID

NCT04675944

Start Date

February 28 2018

End Date

May 25 2018

Last Update

December 19 2020

Active Locations (1)

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PAREXEL International - Early Phase Clinical Unit

Berlin, Germany, 14050